Glutathione | Compounded Injectable
Glutathione is a naturally occurring antioxidant produced in the body and often referred to as the body’s primary cellular protector. It is composed of three amino acids and plays a role in supporting detoxification pathways, immune health, and protection against oxidative stress. Glutathione also participates in mitochondrial function and helps recycle other antioxidants such as vitamins C and E.
Glutathione levels may decline with age, chronic stress, environmental exposures, or certain medical conditions. Compounded injectable glutathione is prescribed to support antioxidant activity, liver function, and overall cellular health. Your Superior provider will determine if this therapy is appropriate based on your symptoms, medical history, and laboratory findings. Dosing and frequency are individualized and monitored for safety.
This is a compounded injectable formulation dispensed by a licensed compounding pharmacy. Compounded medications are not FDA-approved and have not been reviewed for safety or efficacy. Review important medication safety information.
Important Safety Information: Glutathione 200 mg/mL | Compounded Injectable
What is this?
This Important Safety Information summarizes key warnings and precautions for Glutathione 200 mg/mL, a compounded injectable antioxidant formulation. Glutathione is a naturally occurring tripeptide composed of glycine, cysteine, and glutamic acid and plays a role in cellular antioxidant activity and detoxification processes . This compounded injectable formulation has not been reviewed or approved by the U.S. Food and Drug Administration (FDA) for safety or efficacy and should only be used exactly as directed by a licensed healthcare provider. This summary does not include all available information. Always read your medication label and follow your provider’s instructions.
Most Serious Warnings
Product can cause:
Severe allergic reactions, including rash, hives, swelling of the face, lips, tongue, or throat
Bronchospasm or difficulty breathing
Liver or kidney toxicity in rare cases
Neurological symptoms or nervous system toxicity in rare cases
Interactions with certain medications, including chemotherapeutic agents
Compounded glutathione may carry sterility or formulation risks due to limited FDA oversight.
Who Should NOT Take Glutathione
Do not take this medication if you:
Have a known allergy to glutathione or any ingredient in the formulation
Have been advised to avoid antioxidant or detoxification therapies
Are receiving active chemotherapy unless specifically directed by your oncology provider
Have severe uncontrolled liver or kidney disease without provider clearance
Before Taking Glutathione, Tell Your Healthcare Provider if You:
Have asthma or a history of bronchospasm
Have liver or kidney disease
Are undergoing chemotherapy or cancer treatment
Take high doses of acetaminophen, which may affect glutathione levels
Take any prescription, over the counter, or herbal medications
Are pregnant, planning pregnancy, or breastfeeding
Possible Side Effects
Common (mild to moderate):
Redness, pain, itching, or irritation at the injection site
Mild fatigue following infusion
Abdominal cramping
Skin lightening due to changes in melanin production
Serious (seek medical care immediately):
Rash, hives, swelling of the face or throat, difficulty breathing
Trouble breathing due to bronchial constriction
Signs of liver or kidney problems such as unusual fatigue, dark urine, or decreased urination
Neurological symptoms such as confusion or severe weakness
While Taking Glutathione
Tell your healthcare provider immediately if you:
Develop shortness of breath or wheezing
Experience severe fatigue, weakness, or unusual symptoms
Notice significant changes in skin tone
Have new or worsening symptoms
Pregnancy and Breastfeeding
The safety of injectable glutathione during pregnancy or breastfeeding has not been fully established. Use only under medical supervision if your provider determines that potential benefits outweigh risks.
Overdose
Symptoms of glutathione overdose may include:
Severe abdominal cramping
Difficulty breathing or bronchospasm
Signs of organ toxicity
If overdose is suspected, seek emergency medical attention or contact Poison Control immediately.
Missed Dosage
If you miss a scheduled dose:
Do not double the next dose
Follow your provider’s instructions for rescheduling
Contact your provider or pharmacy if you are unsure how to proceed
Storage
Store refrigerated as directed on the pharmacy label
Protect from light
Do not freeze
Keep out of reach of children
Medication Disposal
Dispose of unused or expired medication according to local medication disposal guidelines. Do not flush medication or dispose of it in household drains. Contact your pharmacy for disposal instructions or ask about medication take back programs.
Provider Oversight and Order Review
This compounded medication requires review and oversight by licensed Superior Health & Wellness providers. Dosing, administration route including intravenous or intramuscular use , and treatment schedules must be discussed directly with your provider to ensure safety and clinical appropriateness. Orders may be adjusted based on labs, goals, and response to therapy.
Telemedicine Disclosure
This prescription may be issued via telemedicine. If you experience any concerning or severe symptoms, contact your prescribing clinician immediately or seek emergency medical care.
Disclaimer
This summary does not include all information about Glutathione and should not replace medical guidance. Always consult your healthcare provider or pharmacist for complete safety information, potential interactions, and individualized treatment recommendations. This compounded medication has not been evaluated or approved by the FDA for safety or efficacy.
You are encouraged to report negative side effects of prescription drugs to the FDA. Visit MedWatch or call 1-800-FDA-1088.
